Both Zopiclone 7.5mg and 10mg are prescription medications that help to treat insomnia or sleeplessness in adults. It is intended for only short-term use. It is a sedative hypnotic that works by calming down the brain activity and nervous system. As a result, it helps to fall asleep faster and remain asleep throughout the night.
Doctors usually prescribe Zopiclone 7.5mg & 10mg when other therapeutic and lifestyle changes fails to restore the sleep cycle. They prescribe Zopiclone or other z-drugs when all other alternative remedies fails.
Zopiclone might be an excellent choice for people who struggle to fall asleep fast or suffer from frequent night awakenings. However, it does content certain risks and side-effects that you must be aware of before taking the medicine. Remember, Zopiclone is meant short-term usage. Therefore, taking it for too long can lead to dependency and other serious side effects.
What is Zopiclone 7.5mg & 10mg?
Zopiclone is available in various dosages such as 3.75mg, 7.5mg, 10mg, 11.25mg and so on. However, the most commonly used dosages of Zopiclone are Zopiclone 7.5mg and 10mg. Zopiclone belongs to a group of medicine known as non-benzodiazepine hypnotics. Zopiclone is generally used for the short-term treatment of insomnia.
Zopiclone offers treatment of insomnia by reducing sleep latency or time one takes to fall asleep, increases sleep duration and also reduces the number of night awakenings to promote healthy sleep cycle. The medicine should only be used by adults for a short time (ideally 7-14 days) to treat sleeplessness and other sleep problems.
Mechanism of Action
Zopiclone 7.5mg and 10mg are available as oral tablets. These oral tablets belong to the category of non-benzodiazepine hypnotics. Zopiclone is a fast-acting sleep disorder drug that at most half an hour to 1 hour to start acting after ingestion.
Zopiclone binds with gamma-aminobutyric acid type A or GABAA (a chemical receptor of the brain). GABAA creates a calming effect on the mind. It enhances the effects of GABAA, which has anxiolytic and hypnotic properties. The sedative and hypnotic properties of GABAA is helpful for creating a calming effect on the brain and initiate sleep. It also ensures that a person remains asleep throughout the night (7-8 hours of sleep).
Non-Benzodiazepine Classification
Zopiclone 7.5mg and 10mg are non-benzodiazepine hypnotics that belong to the pyrazolopyrimidine class. It is designed for the short-term treatment of insomnia. The medicine, like other non-benzodiazepine hypnotics, binds with a certain chemical receptor of the brain, GABAA. Zopiclone works by modulating benzodiazepine receptors. Its final aim is to enhance the impact of GABAA on the brain. This helps to relax the nerves in the brain which is helpful for falling asleep faster.
Zopiclone also belongs to a class of medicines known as the ‘Z’ drugs. ‘Z’ are considered powerful non-benzodiazepines that offers effective and quick solutions insomnia and other sleep problems.
Clinical Uses and Indications
Zopiclone 7.5mg and 10mg are generally used for the treatment of insomnia in adults. The medicine is used for short-term treatment. Zopiclone oral tablets are used for these sleep problems:
Treatment of Insomnia
Zopiclone 7.5mg and 10mg are oral sedative-hypnotic tablets. These medicines are used for adult use only. Adults can use this medicine as a short-term treatment option for insomnia. Both Zopiclone 7.5mg and 10mg are used to reduce the symptoms of sleeplessness at night. This medicine reduces sleep latency and facilities faster onset of sleep. It also helps one to stay asleep throughout the night with a reduced number of night awakenings. Zopiclone is also useful for improving the quality of sleep.
Treatment of Frequent Night Awakenings
Frequent nocturnal awakenings can impact the quality of sleep. The medicine enhances the effects of the GABAA receptor and creates a calming effect on the brain. This is particularly helpful for reducing the number of night awakenings and improving overall sleep quality. It also effectively improves sleep duration and ensures 7-8 hours of uninterrupted sleep for improved sleep hygiene. Reducing frequent night awakenings also improves mood and alertness during the daytime.
Treatment of Anxiety-related Sleep Problems
Zopiclone 7.5mg and 10mg are also recommended for anxiety-related sleep problems. Zopiclone binds with the GABAA receptors and also blocks the activities of certain neurotransmitters of the brain. This relaxes the brain nerves and offers relief from the symptoms of anxiety and stress by creating a soothing effect on the mind. This relaxed and calm state of the mind is helpful for sound sleep at night. In some rare cases, the medicine is also used for relieving the symptoms of anxiety. However, this is an off-label use.
Short-Term Use
All the dosages of Zopiclone are designed for short-term use. This medicine can be used for quick relief from the symptoms of insomnia and other sleep problems, such as sleep latency and frequent night awakenings. However, the medicine should be taken for 7-14 days and not more than that. Long-term use of Zopiclone can lead to dependency and withdrawal symptoms.
Comparison to Other Benzodiazepines
Zopiclone belongs to the z-drugs category which is distinctively different from benzodiazepine and other hypnotic drugs. Usually, z-drugs such as Zopiclone tends to be safer and effective along with reduced chances hangover than benzodiazepine class drugs.
Here is a quick comparison of Zopiclone 7.5mg and 10mg with other benzodiazepine class drugs:
| Medicine | Onset | Duration | Common Side Effects |
|---|---|---|---|
| Zopiclone 7.5mg & 10mg | Fast | 6-12 hours | Drowsiness, dizziness and fatigue |
| Lorazepam | Moderate | 8-12 hours | Drowsiness, weakness, unsteadiness |
| Diazepam | Fast | 12-24 hours | Sedation and fatigue, impaired coordination |
While Lorazepam and Diazepam last longer and can be quite beneficial for insomnia issues. They also have higher hangover rates and serious side effects than Zopiclone. On the other hand, Zopiclone 7.5mg and 10mg are safer and more effective for people who struggle with sleeplessness, especially during night time.
Dosage, Administration, and Safety
Zopiclone 7.5mg and 10mg can be a good choice for managing insomnia-like sleep conditions. However, knowing the safety concerns and getting the right dosage is the key to safe and effective usage.
Recommended Dosage
For most adults the recommended dosage is 7.5mg once a day right before bedtime. The dosage can be increased gradually up to 10mg per day for a few days. Remember, Zopiclone is meant for short-term use and may not advisable for more than four weeks.
Also, for elderly adults the dosage can be LS (3.75mg) or full 7.5mg once a day right before bedtime. For these individuals higher dosages often not advisable as they are prone to fall and confusion.
Administration Guidelines
People with serious liver problem must use the medicine with extra caution. Also, children and adolescents under the age of 18 are not recommended to use Zopiclone. Zopiclone works best at night or when you have a long time to complete rest. Therefore, it is advisable to take your oral Zopiclone tablets (as prescribed by your doctor) right before bedtime for optimal results.
Potential Side Effects
Zopiclone has certain side effects common to the z-drugs category, including dry mouth, bitter or metallic taste, nausea, and headache. It also causes a mild sedation or drowsiness that can make it challenging to drive or work with heavy machinery.
For some people it can also cause depression, breathing difficulties and confusion. Allergic reactions are rare with Zopiclone which can cause swollenness, rashes and breathing issues.
Drug Interactions
It is not recommended to take Zopiclone 7.5mg or 10mg with any other sedative or benzodiazepine class drug as it can worsen the side-effects leading to overdosing or misuse. It is also advised not to consume alcohol when taking Zopiclone as it can lead to serious side-effects.
Special Considerations
While taking Zopiclone can be quite beneficial for managing insomnia or sleeplessness. It may not be safe for everyone. People with breathing issues, personality disorders, and anxiety disorder must not use Zopiclone as it can worsen these conditions.
Dependence, Risks, and Precautions
Zopiclone 7.5mg and 10mg are recommended for short-term use. Long-term use of the medicine and overuse can cause dependency and increase the risks of side-effects. People should also take certain precautions to reduce the risks of health hazards while taking Zopiclone.
Signs of Dependence
- Strong and excessive urge to take the medicine
- Need for overdosing on the medicine for more effectiveness
- Finding difficulty falling asleep without the medicine
- Experiencing symptoms of anxiety for not taking the medicine
Precautions
- One should avoid consuming alcohol or other substances that can interact with Zopiclone
- People should also avoid medicines that can interact with Zopiclone
- Pregnant and breastfeeding women should avoid using Zopiclone
- Older adults should not use the strong dosages of Zopiclone such as 7.5mg and 10mg
- People with kidney problems or liver diseases should avoid using Zopiclone
Managing Risks
- Zopiclone 7.5mg and 10mg should be taken for short-term treatment of insomnia.
- Zopiclone 7.5mg and 10mg should only be used by adults experiencing the symptoms of insomnia.
- One should not take Zopiclone every night.
- One should ensure 7-8 hours of uninterrupted sleep after taking the medicine.
- One should take the medicine as prescribed by their healthcare provider, or only one dose of 7.5mg or 10mg in 24 hours. One should not take more than one tablet of Zopiclone in a day.
Zopiclone 7.5mg & 10mg Price
Zopiclone comes in different strengthens such as 3.75mg, 7.5mg and 10mg. The price of the medicine hence vary depending on the strength and pack sizes.
Here’s a look at typical price ranges in the UK:
| Pack Size (Tablets) | Strength | Price Range (GBP) |
|---|---|---|
| 14 | 7.5mg | £12 - £20 |
| 28 | 7.5 mg | £19 - £35 |
| 70 | 10 mg | £94 |
| 140 | 10 mg | £169 |
| 280 | 10mg | €310 |
Prices can vary between pharmacies and might not include delivery fees.
Frequently Asked Questions (FAQ)
What is Zopiclone 7.5mg and 10mg used for?
Zopiclone 7.5mg and 10mg are generally used for the short-term treatment of insomnia. The medicine designed for adult use only. Children and older adults should not use this medicine.
What should one avoid while using Zopiclone?
One should avoid using alcohol and other medications or substances that can interact with Zopiclone 7.5mg or 10mg. Also, one should avoid driving or operating heavy machinery 12hours after taking the medicine.
What are the common side effects of Zopiclone?
Zopiclone 7.5mg and 10mg can cause some minor side effects as your body adjusts to the effects of the medicine. Some common side effects of Zopiclone include dry mouth, metallic taste in the mouth, drowsiness, dizziness, and feelings of confusion.
Can one take Zopiclone every night?
Ideally, Zopiclone 7.5mg or 10mg should not be taken every night. This medicine can be used for 2-3 night every week for at most 2 weeks. Zopiclone should not be used for a long time or regularly.
How long does it take for Zopiclone 7.5mg and 10mg to work?
Both Zopiclone 7.5mg and 10mg act quickly. They have a faster onset time and start working within 1 hour after the ingestion of the medicine.
How long do the effects of Zopiclone last?
The effects of Zopiclone also last longer to ensure longer hours of sleep. The effects of Zopiclone usually last for 12 hours.
